bibonase nasal spray - Uses, Price, Side Effects & Substitutes
What is bibonase nasal spray used for?
Azeflo Nasal Spray (Fluticasone Propionate + Azelastine) is used to treat RESPIRATORY. It contains Fluticasone Propionate (50mcg) + Azelastine (140mcg), which Fluticasone propionate is a corticosteroid that reduces inflammation by inhibiti. Always consult your doctor before use. Take as prescribed.
- Generic Name: Fluticasone Propionate + Azelastine
- Manufacturer: Bibo Pharma
- Form: Allopathy
- Pregnancy Category: C
- Prescription Required: Yes
๐ bibonase nasal spray Uses & Benefits
Seasonal and perennial allergic rhinitis.
Off-label uses: Non-allergic rhinitis; nasal polyps (fluticasone component).
๐ Drug Information
| Generic Name(s) | Fluticasone Propionate + Azelastine |
| Brand Name | Azeflo Nasal Spray |
| Manufacturer | Bibo Pharma |
| Packaging / Form | Varies by brand (Allopathy) |
| Therapeutic Class | RESPIRATORY |
| Action Class | Corticosteroid + Antihistamine |
| Route of Administration | Intranasal |
| Storage | Store at 20-25ยฐC (68-77ยฐF); protect from light. |
| Shelf Life | As per manufacturer |
๐ฌ Pharmacology (PK/PD)
Pharmacokinetics
How It Works
Fluticasone propionate is a corticosteroid that reduces inflammation by inhibiting inflammatory mediators. Azelastine is an antihistamine that blocks histamine H1 receptors, reducing allergic symptoms.
Mechanism Steps
๐ก How to Take bibonase nasal spray
Follow your doctor's prescription exactly.
โ ๏ธ Side Effects of bibonase nasal spray
โ Common Side Effects
- Headache
- Epistaxis
- Nasal discomfort
- Sneezing
- Bitter taste
๐จ Serious Side Effects
- Nasal ulceration
- Perforation
- Glaucoma
- Cataracts
- Adrenal suppression
โ ๏ธ Rare Side Effects
- Anaphylaxis
- Angioedema
- Bronchospasm
Consult your doctor if you experience any unusual symptoms.
๐ฌ Drug Interactions
| โ ๏ธ Drug | Severity | Effect |
|---|---|---|
| Ketoconazole | Major | Increased fluticasone systemic exposure |
| Ritonavir | Major | Increased fluticasone systemic exposure |
| Rifampin | Moderate | Decreased fluticasone efficacy |
| Fluoxetine | Moderate | Increased azelastine levels |
| Alcohol | Minor | Increased sedation |
๐จ Major Interactions
- CYP3A4 inhibitors (e.g., ketoconazole, ritonavir)
- Other corticosteroids (systemic)
โก Moderate Interactions
- CYP3A4 inducers (e.g., rifampin)
- CYP2D6 inhibitors (e.g., fluoxetine)
โน๏ธ Minor Interactions
- Alcohol
- Sedatives
๐ฝ๏ธ Food Interactions
No significant food interactions.
๐ท Alcohol Interaction
May increase sedation risk.
๐ก๏ธ Safety & Warnings
๐ซ Contraindications
Hypersensitivity to any component; untreated nasal infection.
๐ Monitoring Parameters
Nasal symptoms; signs of adrenal suppression with prolonged use.
๐คฑ Lactation Safety
Caution; limited data, but systemic absorption is low.
๐ Overdose Management
No specific antidote; supportive care. Acute overdose unlikely due to low systemic absorption.
โฐ Missed Dose
Take as soon as remembered; if close to next dose, skip missed dose.