bestor 10 tablet - Rosuvastatin (10mg) medicine

bestor 10 tablet - Uses, Price, Side Effects & Substitutes

No reviews yet
๐Ÿญ Biocon ๐Ÿ“ฆ Varies by brand ๐Ÿ’Š Allopathy ๐Ÿ“… Updated: Jun 22, 2026
๐Ÿ“‹ Prescription Required ๐Ÿ’Š Generic Available
Medically Reviewed
Dr. SaathiMed Expert Panel | Jun 22, 2026

What is bestor 10 tablet used for?

Arvast 10 Tablet (Rosuvastatin) is used to treat CARDIAC. It contains Rosuvastatin (10mg), which Competitive inhibitor of HMG-CoA reductase, the rate-limiting enzyme in choleste. Always consult your doctor before use. Take as prescribed.

  • Generic Name: Rosuvastatin
  • Manufacturer: Biocon
  • Form: Allopathy
  • Pregnancy Category: A
  • Prescription Required: Yes
๐Ÿ’ก Did You Know? The first generic medicine was introduced in India in 1970 after the Patents Act was amended.

๐Ÿ’Š bestor 10 tablet Uses & Benefits

Hypercholesterolemia (primary and mixed dyslipidemia), homozygous familial hypercholesterolemia, prevention of cardiovascular events in patients with risk factors.

Off-label uses: Chronic kidney disease, non-alcoholic fatty liver disease, post-transplant hyperlipidemia.

๐Ÿ“‹ Drug Information

Generic Name(s)Rosuvastatin
Brand NameArvast 10 Tablet
ManufacturerBiocon
Packaging / FormVaries by brand (Allopathy)
Therapeutic ClassCARDIAC
Action ClassHMG CoA inhibitors (statins)
Route of AdministrationOral.
StorageStore at 20-25ยฐC (68-77ยฐF); protect from light and moisture.
Shelf LifeAs per manufacturer

๐Ÿ”ฌ Pharmacology (PK/PD)

Pharmacokinetics

AbsorptionAbsorbed rapidly after oral administration; peak plasma concentrations achieved in 3-5 hours. Absolute bioavailability is approximately 20%.
DistributionDistributed extensively to extravascular sites; volume of distribution is about 134 L. Highly bound to plasma proteins.
Protein BindingApproximately 88% bound to plasma proteins, mainly albumin.
MetabolismMinimal metabolism; approximately 10% is metabolized by CYP2C9 to N-desmethyl rosuvastatin, which has 1/6 to 1/2 the activity of the parent compound.
Half-LifeApproximately 19 hours (range 13-20 hours).
ExcretionPrimarily excreted in feces (90%) as unchanged drug and metabolites; renal excretion accounts for about 10%.
BioavailabilityApproximately 20%.
Onset of ActionOnset of lipid-lowering effect occurs within 1 week, with maximal effect seen after 4 weeks.
Peak Plasma Time3-5 hours.
Duration of ActionDuration of action is approximately 24 hours, allowing once-daily dosing.

How It Works

Competitive inhibitor of HMG-CoA reductase, the rate-limiting enzyme in cholesterol biosynthesis, leading to reduced intracellular cholesterol levels and increased LDL receptor expression.

Mechanism Steps

1Rosuvastatin competitively inhibits HMG-CoA reductase, the enzyme that converts HMG-CoA to mevalonate.
2This reduces intracellular cholesterol synthesis in the liver.
3Decreased intracellular cholesterol leads to upregulation of LDL receptors on hepatocyte surface.

๐Ÿ’ก How to Take bestor 10 tablet

Follow your doctor's prescription exactly.

โš ๏ธ Side Effects of bestor 10 tablet

โœ… Common Side Effects

  • Myalgia
  • Headache
  • Nausea
  • Diarrhea
  • Constipation
  • Abdominal pain
  • Asthenia

๐Ÿšจ Serious Side Effects

  • Rhabdomyolysis
  • Myopathy
  • Hepatotoxicity
  • Acute renal failure (secondary to rhabdomyolysis)
  • Hypersensitivity reactions

โš ๏ธ Rare Side Effects

  • Peripheral neuropathy
  • Memory loss
  • Gynecomastia
  • Interstitial lung disease
  • Tendon rupture

Consult your doctor if you experience any unusual symptoms.

๐Ÿ”ฌ Drug Interactions

โš ๏ธ DrugSeverityEffect
Cyclosporine Major Increased rosuvastatin plasma concentration; risk of myopathy/rhabdomyolysis.
Gemfibrozil Major Increased risk of myopathy/rhabdomyolysis.
Warfarin Major Increased INR and bleeding risk.
Fibrates Major Increased risk of myopathy.
Niacin (lipid-lowering doses) Major Increased risk of myopathy/rhabdomyolysis.
Erythromycin Moderate Moderate increase in rosuvastatin levels.
Itraconazole Moderate Moderate increase in rosuvastatin levels.
Ketoconazole Moderate Moderate increase in rosuvastatin levels.
Protease inhibitors Moderate Increased rosuvastatin exposure.
Amiodarone Moderate Possible increased risk of myopathy.
Verapamil Moderate Possible increased rosuvastatin levels.
Digoxin Minor No significant interaction; minor increase in digoxin levels.
Oral contraceptives Minor Minor increase in ethinyl estradiol and norgestrel levels.
Antacids (aluminum/magnesium) Minor Reduced rosuvastatin absorption; separate by 2 hours.
Fenofibrate Minor No significant interaction.

๐Ÿšจ Major Interactions

  • Cyclosporine
  • Gemfibrozil
  • Warfarin
  • Fibrates
  • Niacin (lipid-lowering doses)

โšก Moderate Interactions

  • Erythromycin
  • Itraconazole
  • Ketoconazole
  • Protease inhibitors
  • Amiodarone
  • Verapamil

โ„น๏ธ Minor Interactions

  • Digoxin
  • Oral contraceptives
  • Antacids (aluminum/magnesium)
  • Fenofibrate

๐Ÿฝ๏ธ Food Interactions

Grapefruit juice may increase rosuvastatin exposure; avoid large quantities. Food does not affect absorption.

๐Ÿท Alcohol Interaction

Alcohol may increase risk of hepatotoxicity; limit consumption.

๐Ÿ›ก๏ธ Safety & Warnings

๐Ÿšซ Contraindications

Active liver disease, unexplained persistent elevations of serum transaminases, pregnancy, lactation, hypersensitivity to rosuvastatin.

๐Ÿ“Š Monitoring Parameters

Lipid profile, liver function tests (ALT, AST) at baseline and periodically, creatine kinase if muscle symptoms occur.

๐Ÿคฑ Lactation Safety

Not recommended; excreted in breast milk in animal studies.

๐Ÿ’Š Overdose Management

No specific antidote; symptomatic and supportive care; monitor liver function and CK levels.

โฐ Missed Dose

Take as soon as remembered; if close to next dose, skip missed dose; do not double dose.

๐Ÿ‘จโ€โš•๏ธ Reviewed by Expert

Dr. SaathiMed Expert Panel

MD, PhD - Pharmacology

Reviewed: Jun 22, 2026

๐Ÿ”— View Profile

๐Ÿ”„ Substitutes for bestor 10 tablet

View All

Alternative brands with exact same active ingredient (Rosuvastatin (10mg)):

Medical Note: Always consult your doctor before switching medications.

๐Ÿ˜Š Was this information helpful?

Browse Medicines A-Z

Search our extensive medical database alphabetically.

A B C D E F G H I J K L M N O P Q R S T U V W X Y Z
Back to Medicines Directory
SaathiMed App
SaathiMed App Consult doctors & order medicines faster
Install