amess eye drop - Amikacin (1% w/v) medicine

amess eye drop - Uses, Price, Side Effects & Substitutes

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๐Ÿญ Essential Pharmaceuticals ๐Ÿ“ฆ Varies by brand ๐Ÿ’Š Allopathy ๐Ÿ“… Updated: Jun 23, 2026
๐Ÿ“‹ Prescription Required ๐Ÿ’Š Generic Available
Medically Reviewed
Dr. SaathiMed Expert Panel | Jun 23, 2026

What is amess eye drop used for?

Amikacin Sulphate 500mg Injection (Amikacin) is used to treat OPHTHAL. It contains Amikacin (1% w/v), which Binds to 30S ribosomal subunit, causing misreading of mRNA and inhibition of pro. Always consult your doctor before use. Take as prescribed.

  • Generic Name: Amikacin
  • Manufacturer: Essential Pharmaceuticals
  • Form: Allopathy
  • Pregnancy Category: D
  • Prescription Required: Yes
๐Ÿ’ก Did You Know? Over 80% of the antiretroviral drugs used globally to combat AIDS are supplied by Indian pharmaceutical companies.

๐Ÿ’Š amess eye drop Uses & Benefits

Serious Gram-negative infections (sepsis, pneumonia, complicated UTI, intra-abdominal infections); adjunct in tuberculosis; neonatal sepsis.

Off-label uses: Brucellosis, Plague, Tularemia

๐Ÿ“‹ Drug Information

Generic Name(s)Amikacin
Brand NameAmikacin Sulphate 500mg Injection
ManufacturerEssential Pharmaceuticals
Packaging / FormVaries by brand (Allopathy)
Therapeutic ClassOPHTHAL
Action ClassAminoglycosides
Route of AdministrationIntramuscular, Intravenous
StorageStore at 20-25ยฐC; protect from light; do not freeze.
Shelf LifeAs per manufacturer

๐Ÿ”ฌ Pharmacology (PK/PD)

Pharmacokinetics

AbsorptionRapidly absorbed after intramuscular injection; peak plasma concentrations achieved within 1 hour.
DistributionDistributes widely into extracellular fluids; high concentrations in urine, bile, and synovial fluid; crosses placenta; minimal penetration into cerebrospinal fluid unless meninges inflamed.
Protein Binding0-11%
MetabolismMinimal hepatic metabolism; primarily excreted unchanged.
Half-Life2-3 hours (normal renal function); up to 30-60 hours in renal impairment.
ExcretionRenal excretion (90-98% unchanged) via glomerular filtration.
Bioavailability100% (IM); not absorbed orally.
Onset of ActionRapid (within 1 hour for IM).
Peak Plasma Time1 hour (IM); end of infusion (IV).
Duration of Action8-12 hours (dose-dependent).

How It Works

Binds to 30S ribosomal subunit, causing misreading of mRNA and inhibition of protein synthesis.

Mechanism Steps

1Binds to 30S ribosomal subunit
2Interferes with initiation complex
3Causes misreading of mRNA codons

๐Ÿ’ก How to Take amess eye drop

Follow your doctor's prescription exactly.

โš ๏ธ Side Effects of amess eye drop

โœ… Common Side Effects

  • Nephrotoxicity
  • Ototoxicity (vestibular and cochlear)
  • Nausea
  • Vomiting
  • Rash

๐Ÿšจ Serious Side Effects

  • Acute renal failure
  • Irreversible hearing loss
  • Neuromuscular blockade
  • Anaphylaxis

โš ๏ธ Rare Side Effects

  • Superinfection
  • Clostridium difficile colitis
  • Hypomagnesemia

Consult your doctor if you experience any unusual symptoms.

๐Ÿ”ฌ Drug Interactions

โš ๏ธ DrugSeverityEffect
Neuromuscular blocking agents Major Enhanced neuromuscular blockade, respiratory depression
Cisplatin Major Increased nephrotoxicity and ototoxicity
Loop diuretics Major Increased ototoxicity
Vancomycin Major Increased nephrotoxicity
Penicillins Moderate Synergistic antibacterial effect
NSAIDs Moderate Increased nephrotoxicity risk

๐Ÿšจ Major Interactions

  • Neuromuscular blocking agents
  • Other aminoglycosides
  • Cisplatin
  • Loop diuretics
  • Vancomycin

โšก Moderate Interactions

  • Penicillins (synergy)
  • Cephalosporins
  • NSAIDs
  • Methoxyflurane

โ„น๏ธ Minor Interactions

  • Dimercaprol
  • Indomethacin

๐Ÿฝ๏ธ Food Interactions

No significant food interactions.

๐Ÿท Alcohol Interaction

No known interaction.

๐Ÿ›ก๏ธ Safety & Warnings

๐Ÿšซ Contraindications

Hypersensitivity to amikacin or other aminoglycosides; myasthenia gravis; pre-existing severe renal impairment.

๐Ÿ“Š Monitoring Parameters

Renal function (serum creatinine, BUN), urine output, audiometry, serum drug levels (peak and trough).

๐Ÿคฑ Lactation Safety

Caution; small amounts excreted in breast milk; monitor infant for diarrhea, candidiasis.

๐Ÿ’Š Overdose Management

Supportive care; hemodialysis may enhance elimination; monitor renal function and hearing.

โฐ Missed Dose

Administer as soon as remembered; if near next dose, skip missed dose; do not double dose.

๐Ÿ‘จโ€โš•๏ธ Reviewed by Expert

Dr. SaathiMed Expert Panel

MD, PhD - Pharmacology

Reviewed: Jun 23, 2026

๐Ÿ”— View Profile

๐Ÿ”„ Substitutes for amess eye drop

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Alternative brands with exact same active ingredient (Amikacin (1% w/v)):

Medical Note: Always consult your doctor before switching medications.

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